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THIORPHAN
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DeCS
Descriptor
English
:
Thiorphan
Descriptor
Spanish
:
Tiorfan
Descriptor
Portuguese
:
Tiorfano
Tree Number:
D02.886.030.893
D12.125.166.893
D12.125.481.700.750
Definition
English
:
A potent inhibitor of membrane metalloendopeptidase (ENKEPHALINASE).
Thiorphan
potentiates morphine-induced
ANALGESIA
and attenuates naloxone-precipitated withdrawal
symptoms.
Pharmacological Action:
Protease Inhibitors
History Note
English
:
89
Allowable Qualifiers
English
:
AD
administration & dosage
AE
adverse effects
AG
agonists
AA
analogs & derivatives
AN
analysis
AI
antagonists & inhibitors
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
CT
contraindications
DU
diagnostic use
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Record Number:
23847
Unique Identifier:
D015244
Occurrence in VHL
:
Similar:
DeCS
CID-10
SciELO
LILACS
LIS