Pesquisa sobre: CYTOCHROME P-450 CYP3A 
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Descritor Inglês:   Cytochrome P-450 CYP3A 
Descritor Espanhol:   Citocromo P-450 CYP3A 
Descritor Português:   Citocromo P-450 CYP3A 
Sinônimos Inglês:   CYP3A  
Categoria:   D08.244.453.040.986
D08.811.682.662.582.353
D08.811.682.690.708.170.040.888
D12.776.422.220.453.040.972
Definição Inglês:   A cytochrome P-450 monooxygenase that is involved in an NADPH-dependent electron transport pathway by oxidizing a variety of structurally unrelated compounds, including STEROIDS; FATTY ACIDS; and XENOBIOTICS. This enzyme has clinical significance due to its ability to metabolize a diverse array of clinically important drugs such as CYCLOSPORINE; VERAPAMIL; and MIDAZOLAM. This enzyme also catalyzes the N-demethylation of ERYTHROMYCIN. 
Nota Histórica Inglês:   2006(1980) 
Qualificadores Permitidos Inglês:  
AD administration & dosage AE adverse effects
AN analysis AI antagonists & inhibitors
BI biosynthesis BL blood
CF cerebrospinal fluid CS chemical synthesis
CH chemistry CL classification
CT contraindications DF deficiency
DU diagnostic use DE drug effects
EC economics GE genetics
HI history IM immunology
IP isolation & purification ME metabolism
PK pharmacokinetics PD pharmacology
PH physiology PO poisoning
RE radiation effects SE secretion
ST standards SD supply & distribution
TU therapeutic use TO toxicity
UL ultrastructure UR urine
Número do Registro:   50572 
Identificador Único:   D051544 

Ocorrência na BVS:
 

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